Affinity DataIC50: 24.9nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 34.8nMAssay Description:Inhibition of human ACK1 using EAIYAAPFAKKK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding constant for TNK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Average Binding Constant for ACK1; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding constant for TNK2 kinase domainMore data for this Ligand-Target Pair