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Found 4 Enz. Inhib. hit(s) with Target = 'Adenomatous polyposis coli protein' and Ligand = 'BDBM50369191'
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50369191(CHEMBL4164672)
Affinity DataKd:  210nMAssay Description:Binding affinity to APC (unknown origin) at 37 degC by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50369191(CHEMBL4164672)
Affinity DataKd:  250nMAssay Description:Binding affinity to APC protein (303 to 739 residues) (unknown origin) incubated for 60 mins followed by probe addition and measured after 60 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50369191(CHEMBL4164672)
Affinity DataKd:  220nMAssay Description:Binding affinity to His-tagged APC (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenomatous polyposis coli protein(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50369191(CHEMBL4164672)
Affinity DataKd:  12nMAssay Description:Binding affinity to APC (unknown origin) at 30 degC by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed