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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine kinase' and Ligand = 'BDBM50135900'
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135900(5,6-Diphenyl-7-thiophen-2-yl-pyrido[2,3-d]pyrimidi...)
Affinity DataIC50:  0.550nMAssay Description:Inhibition adenosine kinase activity in rat brain in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50135900(5,6-Diphenyl-7-thiophen-2-yl-pyrido[2,3-d]pyrimidi...)
Affinity DataIC50:  49nMAssay Description:Inhibition of adenosine kinase activity in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed