Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM35785'
TargetAdenosine receptor A1(Homo sapiens (Human))
Vernalis (R+D)

Curated by ChEMBL
LigandPNGBDBM35785(pyrimidine-4-carboxamide, 25)
Affinity DataKi:  122nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Vernalis (R+D)

Curated by ChEMBL
LigandPNGBDBM35785(pyrimidine-4-carboxamide, 25)
Affinity DataKi:  122nM ΔG°:  -38.9kJ/molepH: 7.5 T: 2°CAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed