Affinity DataKi: 100nMAssay Description:Binding affinity at Adenosine A1 receptor in rat brain cortical membrane using [3H]-N6-R-phenylisopropyladenosine (R-PIA) as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 302nMAssay Description:Binding affinity of specific [3H]-R-PIA binding to rat Adenosine A1 receptor in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineChecked by AuthorMore data for this Ligand-Target Pair