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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50263199'
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50263199(CHEMBL4076565)
Affinity DataEC50:  891nMAssay Description:Agonist activity at human A1AR expressed in FlpIn-CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation preincubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50263199(CHEMBL4076565)
Affinity DataEC50:  138nMAssay Description:Agonist activity at human A1AR expressed in FlpIn-CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation preincubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed