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Found 5 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50588460'
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50588460(CHEMBL5187330)
Affinity DataKi:  55nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50588460(CHEMBL5187330)
Affinity DataKi:  141nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50588460(CHEMBL5187330)
Affinity DataKd:  24nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells assessed as kinetic dissociation constant by Nano...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50588460(CHEMBL5187330)
Affinity DataKd:  59nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells assessed as kinetic dissociation constant by Na...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50588460(CHEMBL5187330)
Affinity DataEC50:  0.132nMAssay Description:Agonist activity at human adenosine A1 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed