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Found 6 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM82020'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM82020(1-Methyl-3,9-dihydro-purine-2,6-dione(1-methyl xan...)
Affinity DataKi:  9.00E+3nMAssay Description:Binding of 1 nM [3H]-CHA to Adenosine A1 receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM82020(1-Methyl-3,9-dihydro-purine-2,6-dione(1-methyl xan...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(GUINEA PIG)
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM82020(1-Methyl-3,9-dihydro-purine-2,6-dione(1-methyl xan...)
Affinity DataKi:  1.15E+4nMAssay Description:Affinity against adenosine A1 receptor in the brain membranes by the displacement of [3H]-CPX.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM82020(1-Methyl-3,9-dihydro-purine-2,6-dione(1-methyl xan...)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of 1 nM [3H]- N6- (phenylisopropyl) adenosine binding to Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM82020(1-Methyl-3,9-dihydro-purine-2,6-dione(1-methyl xan...)
Affinity DataKi:  3.60E+4nMAssay Description:Binding affinity to A1 adenosine receptor from rat cortical membrane in presence of [3H]-R-(phenylisopropyl)-adenosineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM82020(1-Methyl-3,9-dihydro-purine-2,6-dione(1-methyl xan...)
Affinity DataKi:  3.60E+4nMAssay Description:Binding affinity at Adenosine A1 receptor in rat brain cortical membrane using [3H]-N6-R-phenylisopropyladenosine (R-PIA) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed