Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM82055'
TargetAdenosine receptor A1(Homo sapiens (Human))
Uppsala University

LigandPNGBDBM82055(3-DEAZAADENOSINE | 9-Deazaado | Adenosine receptor...)
Affinity DataKi:  461nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by PDSP Ki Database
LigandPNGBDBM82055(3-DEAZAADENOSINE | 9-Deazaado | Adenosine receptor...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by PDSP Ki Database
LigandPNGBDBM82055(3-DEAZAADENOSINE | 9-Deazaado | Adenosine receptor...)
Affinity DataKi:  2.15E+4nMAssay Description:Binding affinity to adenosine A1 receptor in rat brain membranes by measuring displacement of specific [3H]PIA as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed