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Found 11 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM85618'
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity against human Adenosine A1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi:  1.20E+3nMAssay Description:Tested for inhibitory activity against human adenosine A1 receptor by displacement of [3H]-DPCPX expressed in CHO cells ; value ranges from 1027-1396More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor expressed in CHO cells; range 1027-1396More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human Adenosine A1 receptor expressed in CHO cells; Range 1030-1400More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed