Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM181013' TargetAdenosine receptor A2a(Homo sapiens (Human))
Sigma-Tau Industrie Farmaceutiche Riunite
US Patent
Sigma-Tau Industrie Farmaceutiche Riunite
US Patent
Affinity DataKi: 22nMpH: 7.4Assay Description:The protein concentration of membrane suspension was determined using the Bradford method (Pierce, Rockford, Ill., USA) with bovine albumin as standa...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Sigma-Tau Industrie Farmaceutiche Riunite
US Patent
Sigma-Tau Industrie Farmaceutiche Riunite
US Patent
Affinity DataKi: 22nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in HEK293 cells after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Sigma-Tau Industrie Farmaceutiche Riunite
US Patent
Sigma-Tau Industrie Farmaceutiche Riunite
US Patent
Affinity DataIC50: 2.30E+3nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in HEK293 cells assessed as inhibition of NECA-induced cAMP accumulation incubated for ...More data for this Ligand-Target Pair
