Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50064697'
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50064697(4-[3-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]-CGS- 21680 from rat striatal membranes Adenosine A2A receptor. Parenthesis indicate 95% confidence limits.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50064697(4-[3-(5-Amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataIC50:  60nMAssay Description:Inhibition of 1 uM NECA-stimulated cyclic AMP levels in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed