Affinity DataKi: 2nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >260nMAssay Description:Binding affinity against Adenosine A2a receptor labeled by [3H]-ZM-241,385 in membranes prepared from HEK-A2A cellsMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2a receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 503nMAssay Description:Binding affinity towards human Adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 503nMAssay Description:Antagonist activity against recombinant human adenosine A2A receptor expressed in HEK-293 cells in presence of [125I]-iodo-ZM241385 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 503nMAssay Description:Antagonist activity against human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 503nMAssay Description:Displacement of [125I]ZM241385 from recombinant human A2A adenosine receptor expressed in HEK293 cell membranes measured after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 503nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 503nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 513nMAssay Description:Binding affinity to recombinant human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 612nMAssay Description:Binding affinity to rat adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 612nMAssay Description:Displacement of [3H]CGS21680 from A2A adenosine receptor in rat striatal membranes measured after 3 hrs in presence of adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 612nMAssay Description:Antagonist activity against adenosine A2A receptor in rat striatal membrane in presence of [3H]-CGS-21,680 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 612nMAssay Description:Binding affinity towards rat Adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 612nMAssay Description:Binding affinity at rat Adenosine A2A receptor by [3H]-CGS- 21680 displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Mus musculus)
Rheinische Friedrich-Wilhelms-Universitat Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universitat Bonn
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]MSX-2 from recombinant mouse A2A adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillatio...More data for this Ligand-Target Pair