Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50125928'
TargetAdenosine receptor A2a(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50125928(2-Furan-2-yl-8-methyl-9-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]- SCH-58261 binding at human Adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50125928(2-Furan-2-yl-8-methyl-9-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  156nMAssay Description:Displacement of [3H]- SCH-58261 binding at human Adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed