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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50173176'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50173176(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50173176(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed