Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50149370'
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50149370(4-Amino-2-(4-methoxy-phenyl)-6-nitro-2H-[1,2,4]tri...)
Affinity DataKi:  47nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50149370(4-Amino-2-(4-methoxy-phenyl)-6-nitro-2H-[1,2,4]tri...)
Affinity DataKi:  47nMAssay Description:Binding affinity against human adenosine A3 receptor expressed in CHO cells by [125I]AB-MECA displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50149370(4-Amino-2-(4-methoxy-phenyl)-6-nitro-2H-[1,2,4]tri...)
Affinity DataKi:  4.33E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed