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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50240839'
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50240839(CHEMBL4062581)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]PSB-11 from human adenosine A3 receptor expressed on CHO cell membranes after 2 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50240839(CHEMBL4062581)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]PSB-11 from human adenosine A3 receptor expressed on CHO cell membranes after 2 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50240839(CHEMBL4062581)
Affinity DataKd:  9.10nMAssay Description:Binding affinity to N-terminal Nano-luc tagged human adenosine A3R expressed in HEK293 cells membraneMore data for this Ligand-Target Pair
In DepthDetails PubMed