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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50518050'
TargetAdenosine receptor A3(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50518050(CHEMBL4464176)
Affinity DataEC50:  0.251nMAssay Description:Agonist activity at human adenosine A3 receptor expressed in FlpIn-CHO cells assessed as inhibition of forskolin-mediated cAMP accumulation preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50518050(CHEMBL4464176)
Affinity DataEC50:  0.158nMAssay Description:Agonist activity at human adenosine A3 receptor expressed in FlpIn-CHO cells assessed as increase in ERK1/2 phosphorylation after 5 mins by alphascre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Shanghaitech University

Curated by ChEMBL
LigandPNGBDBM50518050(CHEMBL4464176)
Affinity DataEC50:  0.0631nMAssay Description:Agonist activity at adenosine A3 receptor (unknown origin) expressed in serum starved CHO cells assessed as increase in cell survival after 24 hrs by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed