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Found 6 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50523419'
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50523419(CHEMBL4462442)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]PSB11 from human A3 adenosine receptor expressed in CHO cell membranes measured after 2 hrs by scintillation spectrometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50523419(CHEMBL4462442)
Affinity DataKi:  525nMAssay Description:Irreversible displacement of [3H]PSB11 from human A3 adenosine receptor expressed in CHO cell membranes measured up to 240 mins by scintillation spec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50523419(CHEMBL4462442)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]PSB11 from human A3 adenosine receptor expressed in CHO cell membranes measured after 0.5 hrs by scintillation spectrometric meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50523419(CHEMBL4462442)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]PSB11 from human A3 adenosine receptor expressed in CHO cell membranes preincubated for 4 hrs followed by [3H]PSB11 addition and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50523419(CHEMBL4462442)
Affinity DataIC50:  794nMAssay Description:Displacement of [3H]PSB11 from human A3 adenosine receptor Y265F (7.36) mutant transiently expressed in CHOK1 cell membranes measured after 2 hrs by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50523419(CHEMBL4462442)
Affinity DataIC50:  1.26E+3nMAssay Description:Displacement of [3H]PSB11 from human A3 adenosine receptor transiently expressed in CHOK1 cell membranes measured after 2 hrs by scintillation spectr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed