TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKi: 132nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity at wild type A3R (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of NECA reduced forskolin stimulated cAMP ...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 257nMAssay Description:Binding affinity to Nluc-A3R (unknown origin) expressed in HEK293 cells by nanoBRET assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens
Curated by ChEMBL
National And Kapodistrian University Of Athens
Curated by ChEMBL
Affinity DataKd: 257nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in Flp-In-CHO cells assessed as dissociation constant by by Schild analysisMore data for this Ligand-Target Pair