Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50591171'
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50591171(CHEMBL5174600)
Affinity DataKi:  65nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50591171(CHEMBL5174600)
Affinity DataIC50:  4.30nMAssay Description:Antagonist activity at wild type A3R (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of NECA reduced forskolin stimulated cAMP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National And Kapodistrian University Of Athens

Curated by ChEMBL
LigandPNGBDBM50591171(CHEMBL5174600)
Affinity DataKd:  302nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in Flp-In-CHO cells assessed as dissociation constant by by Schild analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed