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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50597191'
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50597191(CHEMBL5195631)
Affinity DataKi:  13nMAssay Description:Displacement of CA200645 from NLuc human A3 receptor expressed in HEK293 cells assessed as inhibition constant by NanoBRET binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50597191(CHEMBL5195631)
Affinity DataKd:  55nMAssay Description:Binding affinity to NLuc human A3 receptor expressed in HEK293 cells assessed as dissociation constant by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Cambridge

Curated by ChEMBL
LigandPNGBDBM50597191(CHEMBL5195631)
Affinity DataEC50:  16nMAssay Description:Antagonist activity at human wild type A3R expressed in Flp-In-CHO cells assessed as inhibition of forskolin/ NECA-stimulated cAMP accumulation by me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed