Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Aldo-keto reductase family 1 member C3' and Ligand = 'BDBM50362836'
TargetAldo-keto reductase family 1 member C3(Human)
Gifu Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362836BDBM50362836(ARTEPILLIN)
Affinity DataKi:  680nMAssay Description:Noncompetitive inhibition of human recombinant AKR1C3 expressed in Escherichia coli JM109 cells using S-tetralol as substrate by fluorometry in prese...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAldo-keto reductase family 1 member C3(Human)
Gifu Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362836BDBM50362836(ARTEPILLIN)
Affinity DataKi:  680nMAssay Description:Competitive inhibition of human recombinant AKR1C3 expressed in Escherichia coli JM109 cells using S-tetralol as substrate by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAldo-keto reductase family 1 member C3(Human)
Gifu Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362836BDBM50362836(ARTEPILLIN)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant AKR1C3 expressed in Escherichia coli JM109 cells using S-tetralol as substrate by fluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed