Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor' and Ligand = 'BDBM50005127'
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Predix Pharmaceuticals
Curated by ChEMBL
Predix Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 229nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1 receptor in rat cerebral cortex cellsMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataKi: 229nMAssay Description:Binding affinity to human adrenergic receptor alpha1More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair