Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor' and Ligand = 'BDBM50070101'
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070101BDBM50070101(CHEMBL3407840)
Affinity DataKi:  537nMAssay Description:Displacement of [3H]-RX-821002 from human alpha-2 adrenergic receptor in brain prefrontal cortex membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2016
Entry Details Article
PubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Human)
Trinity College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070101BDBM50070101(CHEMBL3407840)
Affinity DataEC50:  3.57E+3nMAssay Description:Antagonist activity at human alpha-2 adrenergic receptor in brain prefrontal cortex membrane assessed as inhibition of UK14304-induced [35S]-GTPgamma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2016
Entry Details Article
PubMed