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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-2A adrenergic receptor' and Ligand = 'BDBM50412258'
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50412258(CHEMBL451229)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]RS79948-197 from human recombinant adrenergic alpha2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412258(CHEMBL451229)
Affinity DataEC50:  79nMAssay Description:Agonist activity at human recombinant adrenergic alpha2A receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed