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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-2A adrenergic receptor' and Ligand = 'BDBM50476178'
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50476178(CHEMBL223829)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]RX821002 from human adrenergic alpha2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50476178(CHEMBL223829)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human adrenergic alpha-2A receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed