Affinity DataKi: 214nMAssay Description:Displacement of [3H]RX821002 from human adrenergic alpha-2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human adrenergic alpha-2B receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair