Affinity DataKi: 25nMAssay Description:Inhibitory constant determined using [3H]rauwolscine in LM(tk-) cells stably transfected with cloned human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Alpha-2C adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair