Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Amyloid-beta precursor protein' and Ligand = 'BDBM50490495'
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50490495(CHEMBL2326893)
Affinity DataKi:  353nMAssay Description:Displacement of [125I]IMPY from amyloid beta (1 to 42) (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50490495(CHEMBL2326893)
Affinity DataKd:  48nMAssay Description:Binding affinity to amyloid beta aggregate (unknown origin) by centrifugation methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed