TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]DHT from human androgen receptor in MDA453 cellsMore data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at Androgen receptor (unknown origin) transfected in mouse C2C12 cells measured by luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 11.9nMAssay Description:Agonist activity at androgen receptor in mouse C2C12 cells by receptor transactivation assayMore data for this Ligand-Target Pair