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Found 2 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50469103'
TargetAndrogen receptor(Homo sapiens (Human))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50469103(CHEMBL4283232)
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at AR in human LNCAP cells assessed as reduction in DHT-induced transcriptional activation after 24 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50469103(CHEMBL4283232)
Affinity DataIC50:  4.87E+3nMAssay Description:Antagonist activity at AR in human LNCAP cells assessed as reduction in DHT-induced cell growth treated for every 2 days for 4 days by hemocytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed