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Found 2 Enz. Inhib. hit(s) with Target = 'Apelin' and Ligand = 'BDBM50009575'
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Rattus norvegicus)
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataIC50:  1.40nMAssay Description:Agonist activity at rat apelin receptor expressed in CHO cell membranes coexpressing EGFP assessed as inhibition of forskolin-induced cAMP production...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed