Found 4 Enz. Inhib. hit(s) with Target = 'Apelin receptor' and Ligand = 'BDBM50244579' 
Affinity DataKi: 0.150nMAssay Description:Displacement of [125I]-[Nle75, Tyr77] Pyr1-apelin-13 from YFP-tagged human APJ receptor expressed in HEK293 cell membranes after 1 hr by gamma-counti...More data for this Ligand-Target Pair
Affinity DataEC50: 57nMAssay Description:Activity at GFP10-tagged human APJ receptor expressed in HEK293 cells assessed as induction of RlucII-tagged beta-arrestin-2 recruitment after 30 min...More data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Binding affinity against sigma receptor from guinea pig brain (minus cerebellum) homogenates, using the novel [3H]-(+/-)-4 as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Binding affinity against sigma receptor from guinea pig brain (minus cerebellum) homogenates, using [3H]ditolylguanidine (DTG) as radioligand.More data for this Ligand-Target Pair
