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Found 3 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM50345657'
TargetAromatase(Homo sapiens (Human))
University Of Chieti 'G. D'Annunzio

Curated by ChEMBL
LigandPNGBDBM50345657(CHEMBL1784801 | rac-3-((1H-imidazol-1-yl)methyl)-1...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Chieti 'G. D'Annunzio

Curated by ChEMBL
LigandPNGBDBM50345657(CHEMBL1784801 | rac-3-((1H-imidazol-1-yl)methyl)-1...)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of human recombinant aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Chieti 'G. D'Annunzio

Curated by ChEMBL
LigandPNGBDBM50345657(CHEMBL1784801 | rac-3-((1H-imidazol-1-yl)methyl)-1...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of human aromatase assessed as reduction in fluorescence intensity using 7-methoxy-4-trifluoromethyl coumarin as a substrate by fluorimetr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed