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Found 13 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM50398447'
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataKi:  0.950nMAssay Description:Binding affinity to aromatase (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataKi:  10nMAssay Description:Competitive inhibition of human aromatase extracted from placental microsomesMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataKi:  26nMAssay Description:Irreversible inhibition of human aromatase extracted from placental microsomesMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataKi:  26nMAssay Description:Inhibition of human placental microsome aromatase using [3H]androstenedione as substrate preincubated for 32 mins in presence of NADPH followed by su...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataKi:  26nMAssay Description:Competitive inhibition of human placental microsome aromatase using varying levels of [1beta2beta3H]-androstenedione as substrateMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  15nMAssay Description:Inhibition of aromatase in human breast tumorMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  23nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  43nMAssay Description:Inhibition of purified HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  50nMAssay Description:Inhibition of human placental microsome aromatase using [1beta-3H] androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  50nMAssay Description:Inhibition of aromatase in human JEG-3 cells using Androst-4-ene-3,17-dione as substrate incubated for 1 hr and measured by BCA assayMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  50.1nMAssay Description:Inhibition of human placental aromatase using [3H]-1beta-androstenedione as substrate after 16 hrs by [3H]-water methodMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  230nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  900nMAssay Description:Inhibition of human placental microsome aromatase expressed in human MCF7 cells using [1beta-3H] androstenedione as substrate after 1 hr by liquid sc...More data for this Ligand-Target Pair