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Report error Found 3 Enz. Inhib. hit(s) with Target = 'B1 bradykinin receptor' and Ligand = 'BDBM50165843'
TargetB1 bradykinin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50165843(4'-{[3-(3,3,3-Trifluoro-propionylamino)-pyridin-2-...)
Affinity DataKi:  11.8nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50165843(4'-{[3-(3,3,3-Trifluoro-propionylamino)-pyridin-2-...)
Affinity DataKi:  11.8nMAssay Description:Antagonist activity at Bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50165843(4'-{[3-(3,3,3-Trifluoro-propionylamino)-pyridin-2-...)
Affinity DataKi:  12nMAssay Description:Inhibitory constant against human Bradykinin receptor B1 expressed in chinese hamster ovary cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed