Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in clone CHO-D-/aequorin cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHO-D cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Antagonist activity at human bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Antagonistic activity at human bradykinin B1 receptor expressed in CHO cells assessed as effect on DAK-mediated calcium mobilizationMore data for this Ligand-Target Pair