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Found 4 Enz. Inhib. hit(s) with Target = 'B1 bradykinin receptor' and Ligand = 'BDBM50209720'
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50209720((R)-3-(4-fluorophenyl)-N-((R)-7-(pyrrolidin-1-ylme...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHOD cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Amgen

Curated by ChEMBL
LigandPNGBDBM50209720((R)-3-(4-fluorophenyl)-N-((R)-7-(pyrrolidin-1-ylme...)
Affinity DataKi:  151nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50209720((R)-3-(4-fluorophenyl)-N-((R)-7-(pyrrolidin-1-ylme...)
Affinity DataIC50:  19.7nMAssay Description:Antagonist activity at human bradykinin B1 receptor expressed in CHOD cellsassessed as effect on DAK-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Oryctolagus cuniculus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50209720((R)-3-(4-fluorophenyl)-N-((R)-7-(pyrrolidin-1-ylme...)
Affinity DataIC50:  451nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed