Affinity DataKi: 14nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHOD cellsMore data for this Ligand-Target Pair
Affinity DataKi: 208nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 17.4nMAssay Description:Antagonist activity at human bradykinin B1 receptor expressed in CHOD cellsassessed as effect on DAK-induced calcium fluxMore data for this Ligand-Target Pair
Affinity DataIC50: 1.69E+3nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptorMore data for this Ligand-Target Pair