Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHOD cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 127nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at human bradykinin B1 receptor expressed in CHOD cellsassessed as effect on DAK-induced calcium fluxMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at human bradykinin B1 receptor expressed in CHO cells assessed as inhibition of agonist-induced calcium efflux by aquerin based ...More data for this Ligand-Target Pair
Affinity DataIC50: 10.4nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptorMore data for this Ligand-Target Pair