Affinity DataKi: 4.10nMAssay Description:Antagonist activity at human B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in clone CHO-D-/aequorin cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Antagonist activity at human bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11.2nMAssay Description:Antagonist activity at rabbit bradykinin B1 receptor expressed in clone CHO-D-/aequorin cells by aquerin based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11.2nMAssay Description:Inhibition of rabbit B1 receptor by cellular calcium flux assayMore data for this Ligand-Target Pair