Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'B2 bradykinin receptor' and Ligand = 'BDBM50074986'
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074986((E)-N-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-y...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074986((E)-N-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-y...)
Affinity DataIC50:  0.300nMAssay Description:Displacement of [3H]bradykinin from guinea pig B2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074986((E)-N-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-y...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Cavia porcellus)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074986((E)-N-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-y...)
Affinity DataEC50:  56nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed