Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'B2 bradykinin receptor' and Ligand = 'BDBM50074986'
TargetB2 bradykinin receptor(Guinea pig)
Jerini

Curated by ChEMBL
LigandPNGBDBM50074986(N-(2-((4-chloro-2-cyano-3-((2-methylquinolin-8-ylo...)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]bradykinin from guinea pig B2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Jerini

Curated by ChEMBL
LigandPNGBDBM50074986(N-(2-((4-chloro-2-cyano-3-((2-methylquinolin-8-ylo...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of specific binding of [3H]BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Jerini

Curated by ChEMBL
LigandPNGBDBM50074986(N-(2-((4-chloro-2-cyano-3-((2-methylquinolin-8-ylo...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Jerini

Curated by ChEMBL
LigandPNGBDBM50074986(N-(2-((4-chloro-2-cyano-3-((2-methylquinolin-8-ylo...)
Affinity DataEC50:  56nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed