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Found 3 Enz. Inhib. hit(s) with Target = 'BTB/POZ domain-containing protein KCTD12' and Ligand = 'BDBM50505514'
TargetBTB/POZ domain-containing protein KCTD12(Homo sapiens)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50505514(CHEMBL4538754)
Affinity DataKi:  1.43E+3nMAssay Description:Displacement of TAMRA-AAG-SLQLPILHHAYLPSIGGV from recombinant human 6X His-tagged KCTD12 T1 domain (27 to 131 residues) expressed in Escherichia coli...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBTB/POZ domain-containing protein KCTD12(Homo sapiens)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50505514(CHEMBL4538754)
Affinity DataIC50:  6.64E+3nMAssay Description:Displacement of TAMRA-AAG-SLQLPILHHAYLPSIGGV from recombinant human 6X His-tagged KCTD12 T1 domain (27 to 131 residues) expressed in Escherichia coli...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBTB/POZ domain-containing protein KCTD12(Homo sapiens)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50505514(CHEMBL4538754)
Affinity DataEC50:  250nMAssay Description:Binding affinity to recombinant human 6X His-tagged KCTD12 T1 domain (27 to 131 residues) expressed in Escherichia coli BL21 DE3 cells preincubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed