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Found 2 Enz. Inhib. hit(s) with Target = 'BTB/POZ domain-containing protein KCTD12' and Ligand = 'BDBM50505539'
TargetBTB/POZ domain-containing protein KCTD12(Homo sapiens)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50505539(CHEMBL4468344)
Affinity DataKi:  1.36E+4nMAssay Description:Displacement of TAMRA-AAG-SLQLPILHHAYLPSIGGV from recombinant human 6X His-tagged KCTD12 T1 domain (27 to 131 residues) expressed in Escherichia coli...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBTB/POZ domain-containing protein KCTD12(Homo sapiens)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50505539(CHEMBL4468344)
Affinity DataKd:  687nMAssay Description:Binding affinity to recombinant human 6X His-tagged KCTD12 T1 domain (27 to 131 residues) expressed in Escherichia coli BL21 DE3 cells assessed as di...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed