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Found 3 Enz. Inhib. hit(s) with Target = 'Beta-2 adrenergic receptor' and Ligand = 'BDBM50186613'
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50186613(4-hydroxymethyl-2-oxy-furazan-3-carboxylic acid am...)
Affinity DataEC50:  6.30E+3nMAssay Description:Vasodilating activity against phenylephrine-induced contractions in rat thoracic aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50186613(4-hydroxymethyl-2-oxy-furazan-3-carboxylic acid am...)
Affinity DataEC50:  8.60E+4nMAssay Description:Agonist activity at adrenergic beta2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contraction in prese...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50186613(4-hydroxymethyl-2-oxy-furazan-3-carboxylic acid am...)
Affinity DataEC50:  8.60E+4nMAssay Description:Agonist activity at adrenergic beta-2 receptor in guinea pig tracheal rings assessed as myorelaxing activity on carbachol-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed