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Found 3 Enz. Inhib. hit(s) with Target = 'Beta-3 adrenergic receptor' and Ligand = 'BDBM50108088'
TargetBeta-3 adrenergic receptor(Rattus norvegicus)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50108088(CHEMBL3601305)
Affinity DataEC50:  535nMAssay Description:Agonist activity at rat beta3-adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50108088(CHEMBL3601305)
Affinity DataEC50:  13nMAssay Description:Agonist activity at recombinant human beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50108088(CHEMBL3601305)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human recombinant beta3-adrenergic receptor expressed in CHO cells assessed as increase of cAMP level after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed