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Found 2 Enz. Inhib. hit(s) with Target = 'Beta-3 adrenergic receptor' and Ligand = 'BDBM50218165'
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218165((R)-1-(pyridin-3-yl)-2-(2-(4-(thiazol-4-yl)phenoxy...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218165((R)-1-(pyridin-3-yl)-2-(2-(4-(thiazol-4-yl)phenoxy...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at rat adrenergic beta-3 receptor assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed