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Found
1
Enz. Inhib. hit(s) with Target = 'Beta-lactamase TEM' and Ligand = 'BDBM466977'
Target
Beta-lactamase TEM
(Escherichia coli)
Entasis Therapeutics
US Patent
Ligand
BDBM466977
(2-[[(2S,5R)-2-(5-carbamoyl-1,3,4-oxadiazol-2-yl)-3...)
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Affinity Data
IC50: 24nM
Assay Description:
A buffer consisting of 0.1 M sodium phosphate (pH 7.0), 10 mM NaHCO3, and 0.005% Triton X-100 was used for all enzymes. The chromogenic substrate nit...
More data for this Ligand-Target Pair
Target Info
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Ligand Info
PC cid
PC sid
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Details
US Patent
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