Affinity DataKi: 800nMAssay Description:Inhibition constant (Ki) for TEM-1 beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 29.5nMpH: 7.0 T: 2°CAssay Description:The inhibitory concentrations (IC50, [uM]) of the beta -lactamase inhibitors against purified TEM-1, SHV-1 and AmpC beta -lactamases are assessed by ...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Compound was evaluated for beta-lactamase inhibition activity of Escherichia coli after 15 min of preincubation with the enzyme at 37 degree CMore data for this Ligand-Target Pair
Affinity DataIC50: 40.2nMAssay Description:Inhibitory activity against Escherichia coli HA58R Class-III TEM-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of Escherichia coli DH5alpha beta-lactamase TEM-1More data for this Ligand-Target Pair
Affinity DataIC50: 145nMAssay Description:Inhibition of Escherichia coli JT4 beta-lactamase TEM1 assessed as inhibition of nitrocefin hydrolysis preincubated for 5 mins by microtiter plate as...More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of Escherichia coli K12 TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibitory activity against Beta-lactamase type TEM2 (penicillinase) from E. coli TEM2 using penicillin G (40 uM) as a substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:The compound was tested for its inhibitory activity towards Class A TEM-1 beta-lactamase from Escherichia coli at 0.3 umolMore data for this Ligand-Target Pair
Affinity DataIC50: 1.45E+5nMAssay Description:Concentration required for its inhibitory activity against Escherichia coli JT4(TEM1) class A beta-lactamaseMore data for this Ligand-Target Pair